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Description: Restore 90caps by ALRI
Time to Restore?
ALR
Industries Restore is not just another testosterone booster. Though an
increase in testosterone production alone is pretty cool, and one of
the reported major benefits of Restore, it would be only part of the
Restore optimized male matrix. Instead we have opted to see how many
arguments we can start (and knock-offs we can inspire) this time by
raising the bar for product expectations beyond what any one product
can currently offer performance oriented males?by doing the whole job.
Its okay, we are men, we like competition!
Estrogen Control
1.
6-Bromodione: There are two types of estrogen aromatase inhibitors and
application of only one leaves the other pathway open for feminizing
potential.
6 alpha-Bromodione is a competitive inhibitor of
aromatase enzymes. Basically this means it works by way of binding to
the active binding site of the aromatase enzyme resulting in prevention
of interaction with other steroids that aromatize like testosterone and
the rest of our favorite male androgens. This is great for rapid
binding and short term aromatase control, but unfortunately a
competitive inhibitor will eventually let go of the enzyme and allow it
to do feminizing things to manly hormones. So, only half of the job is
done, but it has its important role as well.
2. 6
beta-Bromodione is a mechanism-based irreversible inhibitor of the
aromatase enzyme. An irreversible aromatase inhibitor is also referred
to as a suicide inhibitor. It?s pretty cool in that it acts similar to
a competitive inhibitor in the way it binds, but like a pissed-off
ex-girlfriend, it is both highly selective and it will not let go until
death do they part. Together the two analogs in 6-Bromodione make sure
that estrogen is under control, and many would assume that less
estrogen means the prolactin would be under control as well. Often,
once prolactin increases are stimulated, shutting it back down takes
some extra effort and a protracted period of time. How long are you
willing to wait to be an optimized male?
Prolactin Inhibition
Many
have heard of or used drugs like bromocriptine that inhibit prolactin
production for medical needs. Of course one of the benefits is an often
reported increase in libido, and ?related factors?, but the
side-effects such as nausea and dry mouth can certainly negate the
positive.
Prolact-X (Chasteberry Diterpine Matrix Extract)
There has been a long history of supplemental use of Chasteberry for
treatment of PMS in women. Most researches believe that PMS is commonly
the result of high prolactin levels so no surprise that we took an
interest in this herb.
The
amino acid dopamine is the body?s natural controller of prolactin
release. Of course many dopaminergic compounds have been noted as
effective treatments for increasing GH secretion as well, which
correlates rather well with optimization in male performance due to the
fact that elevated prolactin results in decreased GH and IGF-1
production.
The search for the prolactin-suppressive principles
in Chasteberry provided a number of compounds with dopaminergic
properties. In short, research showed that they bound to recombinant
dopamine DA2-receptors and suppressed prolactin release from cultivated
lactotrophs as well as in animal experiments. The search for the
chemical identity of the dopaminergic compounds resulted in isolation
of a number of diterpenes of which some clerodadienols were most
important for the prolactin-suppressive effects. They were almost more
effective in their prolactin-suppressive properties than dopamine
itself.
Naturally just crushing up a bunch of Chasteberry is not
likely to do the job, but proper preparation of the de-feminizing herb
has finally given us an effective synergist to support male
optimization.
So, cool, now that we have dealt with the HPTA
suppression and feminizing issues. By doing so the obvious result is a
notable and welcomed increase in testosterone production. But hey, why
not push all the way and reach for optimization?
Increased Free Testosterone
Free-T
(Proprietary Pure Avenacosides Matrix)
Seems most males who use supplements for either lean mass gains, libido
augmentation or both have heard of Avena Sativa. Yeah, I know, lots of
products already have some form avena sativa or its extracts in it, so
what makes this one special? Of course we used an extraction process
for maximum active compound content (greatest possible amount of active
milligrams per capsule), but in truth Restore as a product is special,
our Free-T (Proprietary Pure Avenacosides Matrix) from avena sativa
just works well in the whole matrix to provide maximum results.
In
the body testosterone travels around in two forms: Bound or
inactive?meaning it is bound to a protein called SHBGB, and Unbound or
free?meaning it is free to do manly things like build muscle and
increase your capacity to perform sexually.
Basically there are
phytochemicals in avena sativa called avenacosides A and B. Some
studies indicate avenacosides increase actual active or free
testosterone in the body by freeing up the bound testosterone from SHBG
so there is more active testosterone. What good is it to have all kinds
of extra testosterone if it is playing S & M games with SHBG?
Cortisol Inhibition
MbAET
Unless you went coma bound in the early 90?s you have been aware of the
on going benefits reaped and progress made with DHEA and its even
better metabolites. As an example are the patented and effective
products 7-OXO-DHEA and of course 7-Hydroxy-DHEA analogs. Since these
analogs prevent conversion into androgenic metabolites they have been
touted by many as the best thing since pizza. Considering the lack of
androgenic side effects possible while promoting fat loss, lean mass
retention and even maximizing thyroid gland activity, not a real
surprise they have become very popular. Of course oral bioavalability
is pretty poor with most of these analogs thus requiring higher dosages.
Likely
the most powerful and effective DHEA analog is b-AET
(beta-androstenetriol). It has been shown in studies to be between 100
and 100,000 times more active than its DHEA precursor metabolites.
However, like most DHEA analogs there is the issue of poor oral
bioavailability. By supporting the delivery value through simple
alkylation, MbAET is nearly 100% orally bioavailable and only takes a
few milligrams to do its job.
Yeah. I know, get to the fat loss and lean muscle side of things in regard to MbAET?
Glucocorticoids
in humans are in two forms. Inactive cortisone and very active in
eating muscle cortisol. There are two enzymes that are able to make
each of these convert into the other.
11b-HSD-1: Converts
inactive cortisone into cannibalistic cortisol. Studies have implicated
this event in fat tissue as a pathway for increased fat storage. Part
of the reason GH has a positive affect upon body composition is through
its ability to inhibit 11b-HDS-1.
11b-HSD-2: Converts nasty
cortisol into cortisone. 11betaHSD2 debulks intracellular cortisol by
90%. (Let the 11b-HSD-2 rule the house)
Hmmm, so, more 11b-HSD-1 means more cortisol which eats more muscle that likes to help fat do ugly things.
And less 11b-HSD-1 means?
MbAET
inhibits the 11b-HSD-1 enzyme both locally and systemically. This means
that there is less conversion of cortisone to cortisol. Based upon the
studies it appears that in mediating this pathway, it increases immune
function and recovery of cells as well. Less cortisol and fat, more
lean muscle and positive support to health. Not bad!
Optimized Delivery
CYP-X Proprietary Grapefruit Extract)
There
were several studies some years back that showed a dramatic increase in
absorption for some compounds when taken with grapefruit juice. The
reason was due to a specific part of grapefruit called
dihydoxybergamottin (DHB). It decreases the gastronomical destruction
of compounds susceptible to the CYP-450 enzyme thus allowing a far
greater amount of the compound to pass into the body?s circulatory
system instead of the toilet. The components of Restore are a good
example?
By creating an ultra pure active extract of
dihydoxybergamottin (DHB) called CYP-X we have maximally increased the
overall oral bioavailability of our synergistic compounds in Restore
to allow both results and cost effective value in one product.
Don?t Settle?
Having
anything less than optimal testosterone levels is unacceptable for any
male wanting to be the best they can be in all things male, but as a
man excess estrogen and cortisol is a bitch. Restore from ALR
Industries is the newest complete synergistic weapon in the fight
against mediocrity for all men.
Restore is a great product for anyone wanting to be an optimized male. Restore also stacks extremely well with Jungle Warfare
Restore Suggested Use:
As a dietary supplement take one capsule three times daily with meals.
After eight weeks of continuous use, discontinue use for four weeks. Do
not exceed eight weeks of continuous use.
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